Otenabant
A potent, and selective CB1 receptor antagonist with Ki of 0.7 nM/0.12 nM in binding and functional assays respectively; has low affinity (Ki=7600 nM) for human CB2 receptors; reverses cannabinoid agonist mediated responses, reduces food intake, and increases energy expenditure and fat oxidation in rodents.Obesity Phase 3 Discontinued.
Product Specifications
CAS Number
686344-29-6
Product Name Alternative
CP 945598 | CP-945598 | CP945598
Purity
>98% (HPLC)
Solubility
10 mM in DMSO
Smiles
CCNC1 (CCN (CC1) C2=NC=NC3=C2N=C (N3C4=CC=C (C=C4) Cl) C5=CC=CC=C5Cl) C (=O) N
Molecular Formula
C25H25Cl2N7O
Molecular Weight
510.4183
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
4-Piperidinecarboxamide, 1-[8- (2-chlorophenyl) -9- (4-chlorophenyl) -9H-purin-6-yl]-4- (ethylamino) -
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