S1RA
A potent and selective sigma-1 receptor antagonist with Ki of 17 nM; shows excellent selectivity over sigma-2 receptor (Ki>1 uM) ; shows high activity in the mouse capsaicin model of neurogenic pain, exerts dose-dependent antinociceptive effects in several neuropathic pain models.Pain Phase 2 Clinical.
Product Specifications
CAS Number
878141-96-9
Product Name Alternative
E-52862
Purity
>98% (HPLC)
Solubility
10 mM in DMSO
Smiles
CC1=CC (OCCN2CCOCC2) =NN1C1=CC2=CC=CC=C2C=C1
Molecular Formula
C20H23N3O2
Molecular Weight
337.4155
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
Morpholine, 4-[2-[[5-methyl-1- (2-naphthalenyl) -1H-pyrazol-3-yl]oxy]ethyl]-
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