What is the catalog number for Cilomilast?

The catalog number for Cilomilast is orb1300763.

What sizes are available for Cilomilast?

Cilomilast is available in the following size(s): 5 mg, 1 ml x 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg.

How many pack sizes does Cilomilast come in?

Cilomilast is available in 6 different pack sizes.

Is Cilomilast in stock?

Cilomilast is currently made to order / not held in immediate stock. Contact us for lead time.

Cilomilast

Cilomilast (SB-207499) is a selective PDE4 inhibitor with an IC50 of approximately 110 nM, exhibiting potent anti-inflammatory effects with minimal CNS penetration. It has been investigated in clinical Phase 3 trials for chronic obstructive pulmonary disease (COPD) and studied in models of inflammatory cell activation.

Product Specifications

CAS Number

153259-65-5

Product Name Alternative

COPD, chronic, Cilomilast, disease, anti-inflammatory, Ariflo, asthma, HPDE4, obstructive, LPDE4, PDE4, immunomodulatory, Inhibitor, inhibit, phosphodiesterase, Phosphodiesterase, Phosphodiesterase (PDE), SB 207499, SB207499, SB-207499, pulmonary

Field of Research

Metabolism Research

Purity

97.37% (May vary between batches)

Solubility

H2O:< 1 mg/mL (insoluble or slightly soluble) ; DMSO:60 mg/mL (174.71 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:2 mg/mL (5.82 mM) ; Ethanol:31 mg/mL (90.27 mM)