ERK5-IN-2
ERK5-IN-2 is a selective, orally bioavailable ERK5 inhibitor with sub-micromolar potency, exhibiting IC50 values of 0.82 μM against ERK5 and 3 μM for the ERK5-MEF2D complex. This tool compound is used in biochemical and cellular assays to investigate the role of ERK5 signaling in cancer, inflammation, and cardiovascular disease research.
Product Specifications
CAS Number
1888305-96-1
Product Name Alternative
Inhibit, ERK, ERK5IN2, ERK-5-IN-2, ERK5-IN-2, ERK5, ERK5 IN 2, Extracellular signal regulated kinases, Inhibitor
Field of Research
Signal Transduction, Stem Cell & Developmental Biology
Purity
≥95% (May vary between batches)
Solubility
DMSO:10 mg/mL (25.76 mM) ;10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (2.58 mM)
Smiles
Fc1cccc (Br) c1C (=O) c1c[nH]c (c1) C (=O) Nc1cccnc1
Molecular Formula
C17H11BrFN3O2
Molecular Weight
388.19
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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