H4 Receptor antagonist 1
This compound is a potent and selective inverse agonist of the histamine H4 receptor, exhibiting an IC50 of 19 nM. It is a valuable research tool for investigating the role of the H4 receptor in immunological and inflammatory processes, suitable for both in vitro binding assays and in vivo disease model studies.
Product Specifications
CAS Number
848217-00-5
Product Name Alternative
Histamine Receptor, HistamineReceptor, H4 receptor, H4 Receptor antagonist 1, H-4 Receptor antagonist 1, Inhibitor, inhibit
Field of Research
Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery
Purity
98.81% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:1 mg/mL (3.16 mM) ; DMSO:10 mg/mL (31.57 mM)
Smiles
CN1CCN (CC1) c1nc (C) nc2c3cc (Cl) ccc3oc12
Molecular Formula
C16H17ClN4O
Molecular Weight
316.79
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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