Grapiprant
Grapiprant (AAT-007) is a selective EP4 prostaglandin receptor antagonist, exhibiting a Ki of 24 nM for the canine recombinant EP4 receptor. This compound is utilized in research to investigate EP4-mediated pathways in vitro and has been studied in vivo for its potential role in managing pain and inflammation associated with osteoarthritis.
Product Specifications
CAS Number
415903-37-6
Product Name Alternative
CJ-023,423; ARY-007
Field of Research
Immunology & Inflammation, Neuroscience
Purity
>98%
Bioactivity
EP4 receptor antagonist.
Form
Powder
Solubility
Soluble in DMSO (up to at least 10 mg/ml)
Smiles
CCc1nc2c (C) nc (C) cc2n1-c1ccc (CCNC (=O) NS (=O) (=O) c2ccc (C) cc2) cc1
Molecular Formula
C26H29N5O3S
Molecular Weight
491.61
Storage Conditions
-20°C
Notes
For research use only.
Other Product Names
1—[2-[4- (2-Ethyl-4,6-dimethylimidazo[4,5-c]pyridine-1-yl) phenyl]ethyl]-3- (4-methylphenyl) sulfonylurea
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