LLY-507
A potent, selective and cell-active inhibitor of SMYD2 (IC50100-fold selective over a broad range of methyltransferase and non-methyltransferase targets; inhibits SMYD2-mediated methylation of p53 Lys370 and suppresses proliferation of several esophageal, liver, and breast cancer cell lines in a dose-dependent manner (IC50=1.5-6 uM) .
Product Specifications
CAS Number
1793053-37-8
Product Name Alternative
LLY-507 | LLY 507 | LLY507
Purity
>98% (HPLC)
Solubility
DMSO: 15 mg/mL
Smiles
O=C (C1=CC (C2=CC=CC=C2N3CCN (CCN4C=C (C) C5=C4C=CC=C5) CC3) =CC (C#N) =C1) NCCCN6CCCC6
Molecular Formula
C36H42N6O
Molecular Weight
574.7583
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
[1,1'-Biphenyl]-3-carboxamide, 5-cyano-2'-[4-[2- (3-methyl-1H-indol-1-yl) ethyl]-1-piperazinyl]-N-[3- (1-pyrrolidinyl) propyl]-
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