BIX 01294 Trihydrochloride
BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a cell-free assay, reduces H3K9me2 of bulk histones, also weakly inhibits GLP (primarily H3K9me3), no significant activity observed at other histone methyltransferases.
Product Specifications
CAS Number
1392399-03-9
Purity
>98% (HPLC)
Solubility
Ethanol: 8 mg/mL (13.33 mM) ; Water: 98 mg/mL (163.32 mM) ; DMSO: 98 mg/mL (163.32 mM)
Smiles
Cl.Cl.Cl.COC1=C (OC) C=C2C (NC3CCN (CC4=CC=CC=C4) CC3) =NC (=NC2=C1) N1CCCN (C) CC1
Molecular Formula
C28H38N6O2·3HCl
Molecular Weight
600.02
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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