PF 429242
PF-429242 is a competitive inhibitor of sterol regulatory element-binding protein (SREBP) site 1 protease (IC50 = 0.175 μM) . It is selective for site 1 protease against a panel of serine proteases. PF-429242 inhibits rate of cholesterol synthesis in CHO cells (IC50 = 0.53 μM) .
Product Specifications
CAS Number
947303-87-9
Product Name Alternative
PF-429242 | PF 429242 | PF429242
Purity
>98% (HPLC)
Smiles
O=C (c1ccc (CN (CC) CC) cc1) N (CCc1ccccc1OC) [C@@H]1CCNC1.Cl.Cl
Molecular Formula
C25H35N3O2·2HCl
Molecular Weight
482.49
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
(R) -4- ((diethylamino) methyl) -N- (2-methoxyphenethyl) -N- (pyrrolidin-3-yl) benzamide
Available Sizes
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