A922500
A-922500 is a potent orally active inhibitor of DGAT-1 activity, inhibiting both human and mouse forms of the enzymes with IC50 values of 7 and 24 nM, respectively. Acyl CoA/diacylglycerol acyltransferase (DGAT) 1 is one of two known DGAT enzymes that catalyze the final and only committed step in triglyceride biosynthesis.
Product Specifications
CAS Number
959122-11-3
Product Name Alternative
A-922500 | A 922500 | A922500
Purity
>98% (HPLC)
Solubility
DMSO : ≥ 50 mg/mL; 116.69 mM
Smiles
OC (=O) [C@@H]1CCC[C@H]1C (=O) C1=CC=C (C=C1) C1=CC=C (NC (=O) NC2=CC=CC=C2) C=C1
Molecular Formula
C26H24N2O4
Molecular Weight
428.48
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
(1R,2R) -2- (4'- (3-phenylureido) -[1,1'-biphenyl]-4-carbonyl) cyclopentane-1-carboxylic acid
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