PF-3758309
PF-03758309 (IC50=1.3 nM), a pyrrolopyrazole inhibitor of PAK4, has effective ATP-competition.
Product Specifications
CAS Number
898044-15-0
Purity
>98% (HPLC)
Solubility
DMSO : ≥ 100 mg/mL; 203.82 mM
Smiles
CN (C) C[C@@H] (NC (=O) N1Cc2c ([nH]nc2Nc2nc (C) nc3c2scc3) C1 (C) C) c1ccccc1
Molecular Formula
C25H30N8OS
Molecular Weight
490.62
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Available Sizes
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