GSK1016790A
GSK1016790A is a TRPV4 agonist that elicits calcium influx in HEK cells expressing mouse or human TRPV4 (EC50s = 18 and 2.1 nM, respectively) .
Product Specifications
CAS Number
942206-85-1
Product Name Alternative
GSK1016790A | GSK-1016790A | GSK 1016790A.
Purity
>98% (HPLC)
Solubility
DMSO : ≥ 33 mg/mL; 50.33 mM
Smiles
CC (C) C[C@H] (NC (=O) C1=CC2=C (S1) C=CC=C2) C (=O) N1CCN (CC1) C (=O) [C@H] (CO) NS (=O) (=O) C1=C (Cl) C=C (Cl) C=C1
Molecular Formula
C28H32Cl2N4O6S2
Molecular Weight
655.61
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
N-[ (2S) -1-[4-[ (2S) -2-[ (2,4-dichlorophenyl) sulfonylamino]-3-hydroxypropanoyl]piperazin-1-yl]-4-methyl-1-oxopentan-2-yl]-1-benzothiophene-2-carboxamide
Available Sizes
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