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H4 Receptor antagonist 1

H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist with an IC50 of 19 nM.

Product Specifications

CAS Number

848217-00-5

Field of Research

Pharmacology & Drug Discovery

Purity

>98% (HPLC)

Solubility

DMSO:10 mg/mL (31.57 mM)

Smiles

CN1CCN (CC1) c1nc (C) nc2c3cc (Cl) ccc3oc12

Molecular Formula

C16H17ClN4O

Molecular Weight

316.78

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

Available Sizes

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