Relacorilant
Relacorilant is a selective and orally bioavailable antagonist of glucocorticoid receptor (Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively) . Relacorilant has the potential for Cushing’s syndrome treatment.
Product Specifications
CAS Number
1496510-51-0
Product Name Alternative
CORT 125134
Purity
>98% (HPLC)
Solubility
DMSO:10 mM
Smiles
CN1C=C (C=N1) S (=O) (=O) N2CCC3=CC4=C (C[C@@]3 (C2) C (=O) C5=NC=CC (=C5) C (F) (F) F) C=NN4C6=CC=C (C=C6) F
Molecular Formula
C27H22F4N6O3S
Molecular Weight
586.56
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Available Sizes
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