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DY-268

DY-268 is a compound based on trisubstituted pyrazolamide without any FXR agonist activity and cytotoxicity and can be used as an effective FXR antagonist (IC50 = 7.5 nM) .

Product Specifications

CAS Number

1609564-75-1

Purity

>98% (HPLC)

Solubility

DMSO:Soluble; Water: Insoluble

Smiles

Cc (cc1) ccc1-c1nn (Cc2cc (OC) ccc2) cc1C (Nc1cc (S (N2CCOCC2) (=O) =O) c (C) cc1) =O

Molecular Formula

C30H32N4O5S

Molecular Weight

560.66

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

Available Sizes

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