(R) -Elagolix
(R) -Elagolix is a short-acting, nonpeptide, GnRH antagonist with an IC50 and Ki of 0.25 and 3.7 nM, respectively. administered orally, that unlike injectable depot GnRH agonists and antagonists, produces a dose-dependent suppression of ovarian estrogen production, that is, from partial suppression at lower doses to full suppression at higher doses.
Product Specifications
CAS Number
834153-87-6
Product Name Alternative
NBI-56418
Field of Research
Pharmacology & Drug Discovery
Purity
>98% (HPLC)
Solubility
DMSO:100 mg/mL (158.33 mM)
Smiles
CC1=C (C (=O) N (C (=O) N1CC2=C (C=CC=C2F) C (F) (F) F) C[C@@H] (C3=CC=CC=C3) NCCCC (=O) O) C4=C (C (=CC=C4) OC) F
Molecular Formula
C32H30F5N3O5
Molecular Weight
631.59
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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