KPLH1130
KPLH1130 improves glucose tolerance in HFD-fed mice. KPLH1130 is a specific pyruvate dehydrogenase kinase (PDK) inhibitor, blocks macrophage polarization and attenuates proinflammatory responses.
Product Specifications
CAS Number
906669-07-6
Purity
>98% (HPLC)
Solubility
DMSO:130 mg/mL (458.91 mM; Need ultrasonic)
Smiles
O=C1NN=C (C2=CC=C (O) C=C2O) N1C3=CC=C (C) C=C3
Molecular Formula
C15H13N3O3
Molecular Weight
283.28
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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