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KPLH1130

KPLH1130 improves glucose tolerance in HFD-fed mice. KPLH1130 is a specific pyruvate dehydrogenase kinase (PDK) inhibitor, blocks macrophage polarization and attenuates proinflammatory responses.

Product Specifications

CAS Number

906669-07-6

Purity

>98% (HPLC)

Solubility

DMSO:130 mg/mL (458.91 mM; Need ultrasonic)

Smiles

O=C1NN=C (C2=CC=C (O) C=C2O) N1C3=CC=C (C) C=C3

Molecular Formula

C15H13N3O3

Molecular Weight

283.28

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

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