BTSA1.2
BTSA1.2 is a rationalized BTSA1 analog with improved binding to BAX, cellular cytotoxicity, and better toleratence in vivo. Combination of BTSA1.2 with Navitoclax demonstrates synergistic efficacy in apoptosis-resistant cancer cells, xenografts, and patient-derived tumors while sparing healthy tissues.
Product Specifications
CAS Number
2254256-66-9
Purity
>98%
Smiles
O=C1N (N=C (C=2C=CC=CC2) C1N=NC3=NC (=C (S3) C) C) C4=NC (=CS4) C=5C=CC=CC5
Molecular Formula
C23H18N6OS2
Molecular Weight
458.56
Notes
For research use only.
Available Sizes
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