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BTSA1.2

BTSA1.2 is a rationalized BTSA1 analog with improved binding to BAX, cellular cytotoxicity, and better toleratence in vivo. Combination of BTSA1.2 with Navitoclax demonstrates synergistic efficacy in apoptosis-resistant cancer cells, xenografts, and patient-derived tumors while sparing healthy tissues.

Product Specifications

CAS Number

2254256-66-9

Purity

>98%

Smiles

O=C1N (N=C (C=2C=CC=CC2) C1N=NC3=NC (=C (S3) C) C) C4=NC (=CS4) C=5C=CC=CC5

Molecular Formula

C23H18N6OS2

Molecular Weight

458.56

Notes

For research use only.

Available Sizes

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