CPI-0610
CPI-0610 is a small molecule inhibitor of the Bromodomain and Extra-Terminal (BET) family of proteins, with potential antineoplastic activity. Upon administration, the BET inhibitor CPI-0610 binds to the acetylated lysine recognition motifs on the bromodomain of BET proteins, thereby preventing the interaction between the BET proteins and acetylated histone peptides. This disrupts chromatin remodeling and gene expression. Prevention of the expression of certain growth-promoting genes may lead to an inhibition of tumor cell growth.
Product Specifications
CAS Number
1380087-89-7
Purity
>98%
Smiles
ClC1=CC=C (C2=N[C@@] ([H]) (CC (O) =N) C3ON=C (C) C=3C3=CC=CC=C23) C=C1
Molecular Formula
C20H16CLN3O2
Molecular Weight
365.812943458557
Notes
For research use only.
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