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CRT-0066101 hydrochloride

Potent inhibitor of protein kinase D (PKD) ; inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively) .

Product Specifications

CAS Number

1290629-45-6

Smiles

Cl.OC1=CC=C (C2C=NN (C) C=2) C=C1C1=NC=CC (=N1) NC[C@@H] (CC) N

Molecular Formula

C18H23CLN6O

Molecular Weight

374.867821931839

Notes

For research use only.

Available Sizes

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