Cetrorelix
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. (In Vitro) :Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
Product Specifications
CAS Number
145672-81-7
Field of Research
Pharmacology & Drug Discovery
Purity
>98% (HPLC)
Solubility
DMSO:50 mg/mL (33.53 mM)
Smiles
CC (O) =O.CC (C) C[C@H] (NC (=O) [C@@H] (CCCNC (N) =O) NC (=O) [C@H] (Cc1ccc (O) cc1) NC (=O) [C@H] (CO) NC (=O) [C@@H] (Cc1cccnc1) NC (=O) [C@@H] (Cc1ccc (Cl) cc1) NC (=O) [C@@H] (Cc1ccc2ccccc2c1) NC (C) =O) C (=O) N[C@@H] (CCCNC (N) =N) C (=O) N1CCC[C@H]1C (=O) N[C@H] (C) C (N) =O
Molecular Formula
C70H92ClN17O14.C2H4O2
Molecular Weight
1491.11
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Other Product Names
(S) -1- (((R) -2- ((S) -2- ((S) -2- ((R) -2- ((R) -2- ((R) -2-acetamido-3- (naphthalen-2-yl) propanamido) -3- (4-chlorophenyl) propanamido) -3- (pyridin-3-yl) propanamido) -3-hydroxypropanamido) -3- (4-hydroxyphenyl) propanamido) -5-ureidopentanoyl) -L-leucyl-L-arginyl) -N- ((R) -1-amino-1-oxopropan-2-yl) pyrrolidine-2-carboxamide acetate
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