NEO2734
NEO2734 is an orally active and selective inhibitor of p300/CBP and BET bromodomain (IC50 of <30 nM for both p300/CBP and BET bromodomains) .NEO2734, a novel dual inhibitor of BET and CBP/p300, is active in both hotspot mutant (F133V) and non-hotspot mutant (Q165P) PCa cells in vitro and in vivo.
Product Specifications
CAS Number
2081072-29-7
Product Name Alternative
EP31670
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 100 mg/mL (229.65 mM)
Smiles
Cc1cc (cn (C) c1=O) -c1ccc2nc (C3CCOCC3) n (CCOC (F) (F) F) c2c1
Molecular Formula
C22H24F3N3O3
Molecular Weight
435.44
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
Available Sizes
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