GSK620
GSK620 is a pan-BD2 inhibitor, which shows an anti-inflammatory phenotype in human whole blood with excellent broad selectivity, developability, and in vivo oral pharmacokinetics.GSK620 is highly selective for the BET-BD2 family of proteins, with >200-fold selectivity over all other bromodomains. GSK620 shows an anti-inflammatory phenotype in human whole blood.
Product Specifications
CAS Number
2088410-46-0
Purity
>98% (HPLC)
Solubility
DMSO:62.5 mg/mL (192.09 mM; Need ultrasonic)
Smiles
CNC (=O) C1=CC (=CN (C1=O) CC2=CC=CC=C2) C (=O) NC3CC3
Molecular Formula
C18H19N3O3
Molecular Weight
325.4
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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