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ETTAC-2

ETTAC-2 is an LRG1-targeting PROTAC degrader (DC50 = 8.38 μM) that inhibits TGF-β/Smad3 signaling. It reduces pro-fibrotic protein secretion and has been shown in research to slow renal fibrosis progression in experimental models, making it a tool for studying fibrotic diseases.

Product Specifications

Field of Research

Pharmacology & Drug Discovery, Stem Cell & Developmental Biology

Molecular Weight

1891.07

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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