Cathepsin G Inhibitor I
Selected Variant
HY-103351-01
Size: 1 mg
Cathepsin G Inhibitor I (compound 7) is an effective, selective, reversible, competitive, non-peptide cathepsin G inhibitor (IC50=53 nM; Ki=63 nM) [1].
Product Specifications
CAS Number
429676-93-7
UNSPSC
12352005
Target
Cathepsin
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/cathepsin-g-inhibitor-i.html
Concentration
10mM
Purity
99.0
Solubility
DMSO : 50 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C(C1=C(C(N(C2CCN(C(C3=CC=CC=C3)=O)CC2)C)=O)C=C4C=CC=CC4=C1)C(P(O)(O)=O)C5=C6C=CC=CC6=CC=C5
Molecular Formula
C36H33N2O6P
Molecular Weight
620.63
References & Citations
[1]Greco MN, et al. Nonpeptide inhibitors of cathepsin G: optimization of a novel beta-ketophosphonic acid lead by structure-based drug design. J Am Chem Soc. 2002 Apr 17;124 (15) :3810-1.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture and light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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Price
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