Ac-GpYLPQTV-NH2
Ac-GpYLPQTV-NH2 is a STAT3 inhibitor with an IC50 value of 0.33 μM. Ac-GpYLPQTV-NH2 has antitumor activity[1].
Product Specifications
CAS Number
1349616-70-1
UNSPSC
12352209
Target
STAT
Type
Peptides
Related Pathways
JAK/STAT Signaling; Stem Cell/Wnt
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ac-gpylpqtv-nh2.html
Solubility
10 mM in DMSO
Smiles
CC(C)[C@@H](C(N)=O)NC([C@H]([C@H](O)C)NC([C@H](CCC(N)=O)NC([C@H]1N(CCC1)C([C@H](CC(C)C)NC([C@@H](NC(CNC(C)=O)=O)CC2=CC=C(C=C2)OP(O)(O)=O)=O)=O)=O)=O)=O
Molecular Formula
C38H60N9O14P
Molecular Weight
897.91
References & Citations
[1]Uehara Y, et al A. Novel high-throughput screening system for identifying STAT3-SH2 antagonists. Biochem Biophys Res Commun. 2009 Mar 13;380 (3) :627-31.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
STAT3
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