2-Iodomelatonin
2-Iodomelatonin is a potent agonist of melatonin receptor 1 (MT1) with a Ki value of 28 pM, it is more 5-fold selective for MT1 over MT2[1]. 2-iodomelatonin can be used to identify, characterize and localize melatonin binding sites in the brain and peripheral tissues[1].
Product Specifications
CAS Number
[93515-00-5]
UNSPSC
12352005
Target
Melatonin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/2-iodomelatonin.html
Purity
99.04
Solubility
DMF : 30 mg/mL (ultrasonic; warming) |DMSO : 30 mg/mL (ultrasonic; warming) |Ethanol : 20 mg/mL (ultrasonic; warming)
Smiles
CC(NCCC1=C(I)NC2=C1C=C(OC)C=C2)=O
Molecular Formula
C13H15IN2O2
Molecular Weight
358.17
References & Citations
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-101176/2-Iodomelatonin-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-101176/2-Iodomelatonin-SDS-MedChemExpress.pdf
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
MT1
Available Sizes
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