C-7280948
Product Specifications
UNSPSC Description
C-7280948 is a selective and potent protein methyltransferase1 (PRMT1) inhibitor with an IC50 value of 12.75 μM[1].
Target Antigen
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/C-7280948.html
Solubility
DMSO : ≥ 38 mg/mL
Smiles
O=S(C1=CC=C(N)C=C1)(NCCC2=CC=CC=C2)=O
Molecular Weight
276.35
References & Citations
[1]Bissinger EM, et al. Acyl derivatives of p-aminosulfonamides and dapsone as new inhibitors of the arginine methyltransferase hPRMT1. Bioorg Med Chem. 2011 Jun 15;19(12):3717-3731.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-15890/C-7280948-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-15890/C-7280948-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
587850-67-7
Available Sizes
Curated Selection
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