Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

XR9051

XR9051 is an orally active and specific modulator of P-glycoprotein-mediated multidrug resistance (MDR) [1].

Product Specifications

CAS Number

762219-35-2

UNSPSC

12352005

Target

P-glycoprotein

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/xr9051.html

Solubility

10 mM in DMSO

Smiles

O=C(NC1=CC=C(CCN2CC3=C(C=C(OC)C(OC)=C3)CC2)C=C1)C4=CC=CC(/C=C(C(N(C)/C5=C\C6=CC=CC=C6)=O)\NC5=O)=C4

Molecular Formula

C39H38N4O5

Molecular Weight

642.74

References & Citations

[1]I L Dale , et al. Reversal of P-glycoprotein-mediated multidrug resistance by XR9051, a novel diketopiperazine derivative. Br J Cancer. 1998 Oct;78 (7) :885-92.|[2]P Mistry, et al. In vivo efficacy of XR9051, a potent modulator of P-glycoprotein mediated multidrug resistance. Br J Cancer. 1999 Apr;79 (11-12) :1672-8.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Gentamycin-HRP
80-1175 500 ul

Gentamycin-HRP

Sign In for Pricing
View Details
Guanine nucleotide-binding protein subunit beta-like protein Antibody, FITC conjugated
A56357-50UG 50 µg

Guanine nucleotide-binding protein subunit beta-like protein Antibody, FITC conjugated

Sign In for Pricing
View Details
CYP1A1 (Cytochrome P450 1A1, Cytochrome P450-P1, Cytochrome P450 Form 6, Cytochrome P450-C) (HRP)
125561-HRP 100 µL

CYP1A1 (Cytochrome P450 1A1, Cytochrome P450-P1, Cytochrome P450 Form 6, Cytochrome P450-C) (HRP)

Sign In for Pricing
View Details
Gm166 ORF Vector (Mouse) (pORF)
21934014 1.0 µg DNA

Gm166 ORF Vector (Mouse) (pORF)

Sign In for Pricing
View Details
Human Tenascin Protein, His Tag
orb2281248-01 100 µg

Human Tenascin Protein, His Tag

Sign In for Pricing
View Details
Human Tenascin Protein, His Tag
orb2281248-02 1 mg

Human Tenascin Protein, His Tag

Sign In for Pricing
View Details