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PCC16 chloride

PCC16 chloride is a cereblon-based cell-permeable proteolysis-targeting chimera (cp-PROTAC) that degrades the palmitoyltransferase DHHC3 with an IC50 of 102 nM. This compound has shown promising antitumor activity in cellular assays, making it a valuable tool for researching targeted protein degradation in oncology.

Product Specifications

Field of Research

Pharmacology & Drug Discovery

Molecular Weight

4764.69

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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