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TAT-PiET

TAT-PiET is a cell-penetrating peptide inhibitor that disrupts the BRD4/JMJD6 complex by targeting BRD4's ET domain. This inhibition suppresses oncogene expression, impairing breast cancer cell growth in vitro and conferring resistance to endocrine therapy in ERα-positive models, highlighting its research utility in oncology and epigenetics.

Product Specifications

Field of Research

Epigenetics & Chromatin, Signal Transduction

Molecular Weight

2651.07

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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