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JKC363 TFA

JKC363 TFA is a potent and selective melanocortin MC4 receptor antagonist with 90-fold selectivity over MC3 receptors. It inhibits α-MSH-induced TRH release in vitro and demonstrates anti-hyperalgesic effects in vivo, making it a valuable research tool for studying energy homeostasis and pain pathways.

Product Specifications

Field of Research

Immunology & Inflammation, Neuroscience, Pharmacology & Drug Discovery

Molecular Weight

1620.73

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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