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Antileukinate

Antileukinate is an acetylated, amidated hexapeptide antagonist of the CXCR2 chemokine receptor. It blocks IL-8 binding and neutrophil activation in vitro (Ki = 2.7-13 μM) and demonstrates protective effects in vivo, such as reducing acute pancreatitis and associated lung injury in mouse models at 53 mg/kg.

Product Specifications

Field of Research

Cell Biology, Immunology & Inflammation, Pharmacology & Drug Discovery

Molecular Weight

1003.19

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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