Relamorelin acetate

Relamorelin acetate is a potent and selective ghrelin receptor agonist (GHSR, Ki=0.42 nM) that crosses the blood-brain barrier. It stimulates growth hormone release and accelerates gastric emptying, making it a valuable research tool for studying gastroparesis, cachexia, and gastrointestinal motility disorders in both in vitro and in vivo models.