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TAK-448

TAK-448 (MVT-602) is a potent, full kisspeptin receptor (KISS1R) agonist with sub-nanomolar activity (IC50 460 pM; EC50 632 pM) . It has been investigated in preclinical and clinical research for conditions including hypogonadotropic hypogonadism and prostate cancer, exploring its role in modulating the hypothalamic-pituitary-gonadal axis.

Product Specifications

Field of Research

Epigenetics & Chromatin, Pharmacology & Drug Discovery

Molecular Weight

1225.36

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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