CTOP
This small molecule is a potent and selective μ-opioid receptor antagonist (Ki μ=0.96 nM, δ>10,000 nM) . Upon central administration in vivo, it induces behavioral effects. In vitro, it also enhances potassium currents in rat locus coeruleus neurons through a mechanism independent of the μ receptor.
Product Specifications
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Molecular Weight
1062.28
Storage Conditions
-20°C
Notes
For research use only.
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