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Sarafotoxin S6a

This compound is an endothelin receptor agonist, demonstrating potent vasoconstrictive activity in vitro with EC50 values of 7.5 nM in pig coronary artery and >150 nM in guinea pig aorta. It also exhibits nociceptive properties in vivo, making it a useful research tool for studying cardiovascular physiology and pain pathways.

Product Specifications

Field of Research

Pharmacology & Drug Discovery

Molecular Weight

2514.85

Storage Conditions

-20°C

Notes

For research use only.

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