FK 453
Product Specifications
UNSPSC Description
FK 453 (compound 1d) is a potent and selective adenosine A1 receptor antagonist with an IC50 value of 17.2 nM[1].
Target Antigen
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/fk-453.html
Smiles
O=C(/C=C/C1=C2C=CC=CN2N=C1C3=CC=CC=C3)N4[C@@H](CCO)CCCC4
Molecular Weight
375.46
References & Citations
[1]Atsushi Akahane, et al. Discovery of FK453, a novel non-xanthine adenosine A1 receptor antagonist. Bioorganic & Medicinal Chemistry Letters. 1996, 16, 7.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-105275A/FK-453-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-105275A/
Clinical Information
Phase 2
CAS Number
121524-18-3
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
