Dopamine D2 receptor agonist-3
Dopamine D2 receptor agonist-3 (compound 3) is a selective D2 receptor partial agonist and Dopamine D3 receptor antagonist (with pEC50 of 8.3 and [1].
Product Specifications
CAS Number
1257326-24-1
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Dopamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/dopamine-d2-receptor-agonist-3.html
Purity
98.30
Solubility
DMSO : 3 mg/mL (ultrasonic)
Smiles
O=C1N(CC2NCCCC2)CCN1C3=CC=CC=C3.[H]Cl
Molecular Formula
C15H22ClN3O
Molecular Weight
295.81
Precautions
H302, H315, H319, H335
References & Citations
[1]Holmes IP, et al. The identification of a selective dopamine D2 partial agonist, D3 antagonist displaying high levels of brain exposure. Bioorg Med Chem Lett. 2010 Mar 15;20 (6) :2013-6.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
D2 Receptor; D3 Receptor
Available Sizes
Frequently Asked Questions
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