PDK1 allosteric modulator 1
PDK1 allosteric modulator 1 is a molecule targeting PDK1 with a binding affinity of 8 μM. PDK1 allosteric modulator 1 is able to bind to the PIF pocket of PDK1, potentially affecting the biological activity of this kinase[1].
Product Specifications
CAS Number
[303134-93-2]
UNSPSC
12352211
Hazard Statement
H315, H319
Target
PDK-1
Type
Reference compound
Related Pathways
PI3K/Akt/mTOR
Applications
Cancer-Kinase/protease
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/pdk1-allosteric-modulator-1.html
Purity
99.34
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(CN1C(SCCOC2=C(F)C=CC=C2)=NC3=C1C=CC=C3)O
Molecular Formula
C17H15FN2O3S
Molecular Weight
346.38
Precautions
H315, H319
References & Citations
[1]Small-Molecule Allosteric Modulators of the Protein Kinase PDK1 from Structure-Based Docking
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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