GPR40/FFAR1 modulator 1
GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) [1].
Product Specifications
CAS Number
[874755-26-7]
UNSPSC
12352005
Target
Free Fatty Acid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gpr40-ffar1-modulator-1.html
Concentration
10mM
Purity
98.28
Solubility
DMSO : 31.25 mg/mL (ultrasonic)
Smiles
CC1=CC=CC=C1NC2=NC(COC3=CC=C(C(C)=CC(O4)=O)C4=C3)=NC(N)=N2
Molecular Formula
C21H19N5O3
Molecular Weight
389.41
References & Citations
[1]Lückmann M, et al. Molecular dynamics-guided discovery of an ago-allosteric modulator for GPR40/FFAR1. Proc Natl Acad Sci U S A. 2019 Apr 2;116 (14) :7123-7128.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
SC402257 10 µg
MIR6816 Human MicroRNA Expression Plasmid (MI0022661)
Sign In for Pricing
View Details 
TP321254L 1 mg
Tryptophan Hydroxylase (TPH1) (NM_004179) Human Recombinant Protein
Sign In for Pricing
View Details 