GPR40/FFAR1 modulator 1

GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) [1].

Product Specifications

CAS Number

[874755-26-7]

UNSPSC

12352005

Target

Free Fatty Acid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Metabolism-sugar/lipid metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/gpr40-ffar1-modulator-1.html

Concentration

10mM

Purity

98.28

Solubility

DMSO : 31.25 mg/mL (ultrasonic)

Smiles

CC1=CC=CC=C1NC2=NC(COC3=CC=C(C(C)=CC(O4)=O)C4=C3)=NC(N)=N2

Molecular Formula

C21H19N5O3

Molecular Weight

389.41

References & Citations

[1]Lückmann M, et al. Molecular dynamics-guided discovery of an ago-allosteric modulator for GPR40/FFAR1. Proc Natl Acad Sci U S A. 2019 Apr 2;116 (14) :7123-7128.

Shipping Conditions

Room Temperature

Storage Conditions

4°C (Powder, protect from light)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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