Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

CDK8-IN-1

CDK8-IN-1 is a potent and selective CDK8 inhibitor with an IC50 of 3 nM.

Product Specifications

CAS Number

1629633-48-2

UNSPSC

12352005

Target

CDK

Type

Reference compound

Related Pathways

Cell Cycle/DNA Damage

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/CDK8-IN-1.html

Purity

99.77

Solubility

DMSO : 100 mg/mL (ultrasonic)

Smiles

NC(C1=C(C(F)(F)F)C(C2=CC=NC=C2)=CN1)=O

Molecular Formula

C11H8F3N3O

Molecular Weight

255.20

References & Citations

[1]Han X, et al. Discovery of potent and selective CDK8 inhibitors through FBDD approach. Bioorg Med Chem Lett. 2017 Sep 15;27 (18) :4488-4492.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

CDK8

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit
E-CL-H0640-01 24 Tests

Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit

Sign In for Pricing
View Details
Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit
E-CL-H0640-02 48 Tests

Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit

Sign In for Pricing
View Details
Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit
E-CL-H0640-03 96 Tests

Human COL5α2 (Collagen Type V Alpha 2) CLIA Kit

Sign In for Pricing
View Details
ScreenQuest™ Beta-Lactamase Inhibitor Screening Kit
11333-AAT 100 Tests

ScreenQuest™ Beta-Lactamase Inhibitor Screening Kit

Sign In for Pricing
View Details
PE/Cyanine5 Anti-Mouse CD11a Antibody[FD441.8]
E-AB-F1033G-01 50 Tests

PE/Cyanine5 Anti-Mouse CD11a Antibody[FD441.8]

Sign In for Pricing
View Details
PE/Cyanine5 Anti-Mouse CD11a Antibody[FD441.8]
E-AB-F1033G-02 100 Tests

PE/Cyanine5 Anti-Mouse CD11a Antibody[FD441.8]

Sign In for Pricing
View Details