YM471 (free base)
Product Specifications
UNSPSC Description
YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1].
Target Antigen
Endogenous Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/ym471-free-base.html
Smiles
O=C(C1=CC=C(C=C1)NC(C2=C(C3=CC=CC=C3)C=CC=C2)=O)N4C5=CC=CC=C5/C(C(F)(CC4)F)=C/C(N6CCC(CC6)N(C)C)=O
Molecular Weight
648.74
References & Citations
[1]Pharmacological characterization of YM471, a novel potent vasopressin V(1A) and V(2) receptor antagonist
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-116066/YM471-free-base-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-116066/
Clinical Information
No Development Reported
CAS Number
183173-00-4
Curated Selection
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