YM471 (free base)
YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1].
Product Specifications
CAS Number
[183173-00-4]
UNSPSC
12352005
Target
Endogenous Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/ym471-free-base.html
Smiles
O=C(C1=CC=C(C=C1)NC(C2=C(C3=CC=CC=C3)C=CC=C2)=O)N4C5=CC=CC=C5/C(C(F)(CC4)F)=C/C(N6CCC(CC6)N(C)C)=O
Molecular Formula
C39H38F2N4O3
Molecular Weight
648.74
References & Citations
[1]Pharmacological characterization of YM471, a novel potent vasopressin V (1A) and V (2) receptor antagonist
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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