Encaleret
Product Specifications
UNSPSC Description
Encaleret (CLTX-305) is an orally active CaSR antagonist[1].
Target Antigen
CaSR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/encaleret.html
Solubility
DMSO : 350 mg/mL (ultrasonic)
Smiles
O=C(C1=CC=C(C2=CC=CC=C2[C@H](OC[C@H](O)CNC(C)(C)CC3=CC=C(Cl)C(F)=C3)C)C=C1C)O
Molecular Weight
514.03
References & Citations
[1]Discovery of a Potent and Short Acting Oral Calcilytic with a Pulsatile Secretion of Parathyroid Hormone
Publication Date (Web): December 29, 2010 (Letter)
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-14401/Encaleret-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-14401/Encaleret-SDS-MedChemExpress.pdf
Clinical Information
Phase 3
CAS Number
787583-71-5
Available Sizes
Curated Selection
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