BIM-23056
BIM 23056, a linear octapeptide, is a potent sst3 and sst5 somatostatin receptor antagonist with Ki values of 10.8, 5.7, respectively[1].
Product Specifications
CAS Number
150155-61-6
UNSPSC
12352209
Target
Somatostatin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/bim-23056.html
Purity
99.98
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
OC(C=C1)=CC=C1C[C@H](NC([C@@H](NC([C@H](N)CC2=CC=CC=C2)=O)CC3=CC=CC=C3)=O)C(N[C@@H](C(N[C@@H](CCCCN)C(N[C@@H](C(C)C)C(N[C@H](C(N[C@@H](C(N)=O)CC4=CC5=C(C=CC=C5)C=C4)=O)CC6=CC=CC=C6)=O)=O)=O)CC7=CNC8=CC=CC=C78)=O
Molecular Formula
C71H81N11O9
Molecular Weight
1232.47
References & Citations
[1]Y C Patel, et al. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5) . Endocrinology. 1994 Dec;135 (6) :2814-7.|[2]W Feniuk, et al. Further evidence from functional studies for somatostatin receptor heterogeneity in guinea-pig isolated ileum, vas deferens and right atrium. Br J Pharmacol. 1995 Jul;115 (6) :975-80.
Shipping Conditions
Blue Ice
Storage Conditions
-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture)
Scientific Category
Peptides
Clinical Information
No Development Reported
Isoform
SSTR3; SSTR5
Available Sizes
Frequently Asked Questions
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