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Protease-Activated Receptor-2, amide

This synthetic hexapeptide amide (SLIGKV-NH2) acts as a potent agonist for Protease-Activated Receptor-2 (PAR2), with a reported half-maximal inhibitory concentration (IC50) of 10.4 μM. It is widely used in vitro and in vivo to study PAR2-mediated signaling in inflammation, pain, and metabolic research.

Product Specifications

Product Name Alternative

PAR2, inhibit, Inhibitor, Proteaseactivated Receptor, ProteaseactivatedReceptor, ProteaseActivated Receptor2, amide, Protease-Activated Receptor-2, Amide, Protease-Activated Receptor (PAR), Protease Activated Receptor 2, amide, Protease Activated Receptor (PAR), SLIGKV-NH2, Thrombin receptors

Field of Research

Pharmacology & Drug Discovery, Protein Biochemistry

Purity

>99.99% (May vary between batches)

Solubility

H2O:33.33 mg/mL (54.21 mM)

Molecular Weight

614.78

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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