[Lys5, MeLeu9, Nle10]-NKA (4-10)
This compound is a highly selective and potent agonist of the NK2 receptor, exhibiting an IC50 of 6.1 nM. It effectively induces smooth muscle contraction in isolated rat fundus and bladder tissues, with EC50 values of 117 nM and 10 nM, respectively. This makes it a valuable research tool for studying tachykinin receptor function in gastrointestinal and urogenital systems.
Product Specifications
Product Name Alternative
Tachykinin receptor, Neurokinin receptor, Neurokininreceptor, Neurokinin Receptor, NK receptor, NK2, inhibit, Inhibitor, [Lys5, MeLeu9, Nle10] NKA (4 10), [Lys5, MeLeu9, Nle10]-NKA, [Lys5, MeLeu9, Nle10]NKA (410), [Lys-5, MeLeu9, Nle10]-NKA (4-10)
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
>99.99% (May vary between batches)
Solubility
H2O:1 mg/mL (1.24 mM)
Molecular Weight
803.99
Storage Conditions
Keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Notes
For research use only.
Available Sizes
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